General literature
Mechanistic MALDI-TOF Cell-Based Assay for the Discovery of Potent and Specific Fatty Acid Synthase Inhibitors

Weigt D., Parrish CA., Krueger JA., Oleykowski CA., Rendina AR., Hopf C.

Cell Chamical Biology 2019, pii: S2451-9456(19)30205-3. open access

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Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3

Böttcher J., Dilworth D., Reiser U., Neumüller R. A., Schleicher M., Petronczki M., Zeeb M., Mischerikow N., Allali-Hassani A., Szewczyk M. M., Li F., Kennedy S., Vedadi M., Barsyte-Lovejoy D., Brown P. J., Huber K. V. M., Rogers C. M., Wells C. I., Fedorov O., Rumpel K., Zoephel A., Mayer M., Wunberg T., Böse D., Zahn S., Arnhof H., Berger H., Reiser C., Hörmann A., Krammer T., Corcokovic M., Sharps B., Winkler S., Häring D., Cockcroft X. L., Fuchs J. E., Müllauer B., Weiss-Puxbaum A., Gerstberger T., Boehmelt G., Vakoc C. R., Arrowsmith C. H., Pearson M., McConnell D. B.

Nature Chemical Biology 2019, 15 (8), 822–829. open access

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Target 2035: probing the human proteome

Carter AJ., Kraemer O., Zwick M., Mueller-Fahrnow A., Arrowsmith CH., Edwards AM.

Drug Discovery Today 2019, pii: S1359-6446(19)30138-2. open access

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A probe for every protein: Target 2035 — an ambitious open-science proposal to develop a suite of chemical genomics tools to modulate every protein in the proteome — faces many challenges ahead

Mullard A.

Nature Reviews Drug Discovery 2019. open access

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Dectin-1 Is a Marker of Alternatively Activated Macrophages and a Therapeutic Target in Interstitial Fibrotic Lung Diseases

Taweel M. E., Walker H., Mekhael O., Vierhout M., Padwal M., Naiel S., Patel H., Parthasarathy P., Imani J., Ayaub E., Naqvi A., Hirota J. A., Hambly N., Kolb M.R.J., Ask K.

ATS Journals 2019. open access

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An open science rare diseases research initiative: the University of North Carolina Catalyst

Naegeli K., Havener T., Aw W.Y., Anderson E., Morris D.

Future Drug Discovery 2019. open access

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