Success examples
The efflux pump ABCC1/MRP1 constitutively restricts PROTAC sensitivity in cancer cells

Wolf G., Craigon C., Teoh S. T., Essletzbichler P., Onstein S., Cassidy D., Uijttewaal E. C. H., Dvorak V., Cao Y., Bensimon A., Elling U., Ciulli A., Superti-Furga G.

Cell Chem Biol. 2025, 32(2):291-306.e6.