General literature
Designing Effective Lead Molecules against Solid Tumors with Inadequate Treatment Options

Pantsar T.

UNIVERSITY OF EASTERN FINLAND Electronic Publication 2018, ISBN 978-952-61-2748-4. open access.

General literature
Chemically induced degradation of the transcription factor BCL6

Kerres N., Steurer S., Schlager S., Bader G., Berger H., Caligiuri M., Dank C., Engen JR., Ettmayer P., Fischerauer B., Flotzinger G., Gerlach D., Gerstberger T., Gmaschitz T., Greb P., Han B., Heyes E., Iacob RE., Kessler D., Kölle H., Lamarre L., Lancia DR., Lucas S., Mayer M., Mayr K., Mischerikow N., Mück K., Peinsipp C., Petermann O., Reiser U., Rudolph D., Rumpel K., Salomon C., Scharn D., Schnitzer R., Schrenk A., Schweifer N., Thompson D., Traxler E., Varecka R., Voss T., Weiss-Puxbaum A., Winkler S., Zheng X., Zoephel A., Kraut N., McConnell D., Pearson M., Koegl M.

Cancer Research 2017, 20 (12), 2860-2875. open access

Success examples
Mechanistic MALDI-TOF Cell-Based Assay for the Discovery of Potent and Specific Fatty Acid Synthase Inhibitors

Weigt D., Parrish CA., Krueger JA., Oleykowski CA., Rendina AR., Hopf C.

Cell Chemical Biology 2019, 26, 1322-1331 E4. open access

General literature
Mechanistic MALDI-TOF Cell-Based Assay for the Discovery of Potent and Specific Fatty Acid Synthase Inhibitors

Weigt D., Parrish CA., Krueger JA., Oleykowski CA., Rendina AR., Hopf C.

Cell Chamical Biology 2019, pii: S2451-9456(19)30205-3. open access

General literature
Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3

Böttcher J., Dilworth D., Reiser U., Neumüller R. A., Schleicher M., Petronczki M., Zeeb M., Mischerikow N., Allali-Hassani A., Szewczyk M. M., Li F., Kennedy S., Vedadi M., Barsyte-Lovejoy D., Brown P. J., Huber K. V. M., Rogers C. M., Wells C. I., Fedorov O., Rumpel K., Zoephel A., Mayer M., Wunberg T., Böse D., Zahn S., Arnhof H., Berger H., Reiser C., Hörmann A., Krammer T., Corcokovic M., Sharps B., Winkler S., Häring D., Cockcroft X. L., Fuchs J. E., Müllauer B., Weiss-Puxbaum A., Gerstberger T., Boehmelt G., Vakoc C. R., Arrowsmith C. H., Pearson M., McConnell D. B.

Nature Chemical Biology 2019, 15 (8), 822–829. open access

General literature
Target 2035: probing the human proteome

Carter AJ., Kraemer O., Zwick M., Mueller-Fahrnow A., Arrowsmith CH., Edwards AM.

Drug Discovery Today 2019, pii: S1359-6446(19)30138-2. open access